发明名称 |
ПРОИЗВОДНЫЕ) 7-([1, 4]ДИОКСАН-2-ИЛ)БЕНЗОТИАЗОЛА ВКАЧЕСТВЕ ЛИГАНДОВ АДЕНОЗИНОВОГО РЕЦЕПТОРА |
摘要 |
The present invention relates to compounds of the general formula Iwherein R<1>, R<2>, R', R'', n, m and o are defined herein, or a pharmaceutically acceptable salt thereof.It has been found that the compounds of general formula I are adenosine receptor ligands with a good affinity to the A2A-receptor and a high selectivity to the A1- and A3 receptors. These compounds have useful pharmacological activities. |
申请公布号 |
RU2005135154(A) |
申请公布日期 |
2006.06.27 |
申请号 |
RU20050135154 |
申请日期 |
2004.04.07 |
申请人 |
Ф.ХОФФМАНН-ЛЯ РОШ АГ (CH) |
发明人 |
ФЛОР Александер (CH);НОРКРОСС Роджер Дейвид (CH) |
分类号 |
C07D417/14;A61P25/00;C07D417/04;C07D471/08;C07D491/10 |
主分类号 |
C07D417/14 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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