发明名称 BENZISOTHIAZOLE-1, 1-DIOXIDE ACTING AS ANTAGONISTS TO THE VANILLOID RECEPTOR SUBTYPE 1 (VR1) AND USES THEREOF
摘要 <p>Compounds having formula (I) or a pharmaceutically acceptable salt, prodrug, or salt of a prodrug thereof, wherein L, A, G, R&lt;SUP&gt;1&lt;/SUP&gt;, R&lt;SUP&gt;2&lt;/SUP&gt; and R&lt;SUP&gt;3&lt;/SUP&gt; are as defined herein. These compounds are particularly useful in the treatment of pain, inflammatory hyperalgesia, and urinary dysfunctions, such as bladder overactivity and urinary incontinence.</p>
申请公布号 WO2006065646(A1) 申请公布日期 2006.06.22
申请号 WO2005US44613 申请日期 2005.12.07
申请人 ABBOTT LABORATORIES;BROWN, BRIAN, S.;KEDDY, RYAN, G.;LEE, CHIH-HUNG 发明人 BROWN, BRIAN, S.;KEDDY, RYAN, G.;LEE, CHIH-HUNG
分类号 C07D417/04;A61K31/425 主分类号 C07D417/04
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