| 摘要 |
<p>Substituted pyrrolo pyridine compounds (I) and their salts are new. Substituted pyrrolo pyridine compounds of formula (I) and their salts are new. R 1>R-x, -SO 2R-x, -SO 2NR-xR-y, -C(O)OR-x, -C(O)NR-xR-y or tri-1-18C alkylsilyl; R-x, R-y : H, cyclic 1-18C alkyl (optionally substituted), 1-18C alkoxy, 2-6C alkenyl, 4-6C cycloalkenyl, 2-6C alkynyl, 4-24C aryl, 5-18C arylalkyl, 5-18C aryloxy or 5-18C arylalkoxy; R 2>, R 3>H, Cl, F, Br, NO 2, pseudohalogen, formyl (optionally protected), carboxyl, C(S)NH 2, C(O)NH 2, cyclic 1-18C alkyl (optionally substituted), 1-18C fluoroalkyl, 1-18C alkoxy, 1-18C fluoroalkoxy, 2-6C alkenyl, 4-6C cycloalkenyl, 2-6C alkynyl, 4-24C aryl, 5-18C arylalkyl or 5-18C arylalkoxy (where R 3>is 5-18C arylalkyl and it is bonded via the alkyl moiety of the 5-18C arylalkyl radical to the pyridine ring, this alkyl moiety has at least two carbon atoms between aryl moiety of the 5-18C arylalkyl radical or pyridine ring); and X : 1-18C fluoroalkyl. INDEPEDENT CLAIMS are also included for: (1) a mixture comprising one or more (I); (2) the preparation of (I); and (3) a pyrrolo pyridine compounds of formula (VI). Y 1>COR 5>; and R 5>halo, OH or optionally substituted 1-18C alkyloxy, 4-24C aryloxy, or 5-18C arylalkoxy. [Image] [Image].</p> |
