发明名称 |
Acyl derivatives of 5-(2-(4-(1,2 benzaisothiazole-3-yl)-1-piperazinyl)ethyl)-6-chloro-1,3-dihydro-2H-indol-2-one having neuroleptic activity |
摘要 |
A process for preparing acyl derivatives as prodrugs of 5-(2-(4-(1,2 benzisothiazole-3-yl)-1-piperazinyl)ethyl-6-chloro-1,3-dihydro-2H-indol-2-one and pharmaceutically acceptable acid addition salts and methods of use as an antipsychotic. |
申请公布号 |
ZA200502109(B) |
申请公布日期 |
2006.05.31 |
申请号 |
ZA20050002109 |
申请日期 |
2005.03.14 |
申请人 |
PFIZER PRODUCTS INC. |
发明人 |
TIMOTHY NORRIS;ROBERTO COLON-CRUZ |
分类号 |
A61K;A61P;A61P25/18;C07D;C07D417/12 |
主分类号 |
A61K |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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