发明名称 PATENTS USE OF CYSTEINE DERIVATIVES FOR THE PREPARATION OF A MEDICAMENT INTENDED TO TREAT PATHOLOGIES WHICH RESULT FROM THE FORMATION OF THE HETEROTRIMERIC G PROTEIN
摘要 THE INVENTION RELATES TO THE USE OF CYSTEINE DERIVATIVES FOR PREPARING A MEDICAMENT INTENDED TO TREAT DISEASES WHICH RESULT FROM THE FORMATION OF THE HETEROTRIMERIC G PROTEIN. THESE DISEASES INCLUDE IN PARTICULAR DISEASES LINKED TO THE FOLLOWING BIOLOGICAL FUNCTIONS OR DISORDERS: SMELL, TASTE, PERCEPTION OF THE LIGHT, NEUROTRANSMISSION, NEURODEGENERATION, ENDOCRINE AND EXOCRINE GLAND FUNCTIONS, AUTOCRINE AND PARACRINE REGULATION, ARTERIAL TENSION, EMBRYOGENESIS, BENIGN CELL PROLIFERATION, ONCOGENESIS, VIRAL INFECTION, IMMUNOLOGICAL FUNCTIONS, DIABETES, OBESITY, AND BENIGN AND MALIGN PROLIFERATIVE DISEASES. SAID CYSTEINE DERIVATIVES INCLUDE IN PARTICULAR: -BIS-1,L'-[7-(2-AMINO-1-OXO-3-THIOPROPYL)-8-(CYCLOHEXYLMETHYL)-2-(2-METHOXYPHENYL)-5,6,7,8- TETRAHYDROIMIDAZO[1.2A]PYRAZINE DISULPHIDE (I), AND -BIS-1,1'-7-(2-AMINO-1-OXO-3-THIOPROPYL-(2-(1-NAPHTYL)-8-(2-METHYLPROPYL)-5,6,7,8-TETRAHYDROIMIDAZO[1.2A]PYRAZIN-7-YL) DISULPHIDE (II).
申请公布号 MY122419(A) 申请公布日期 2006.04.29
申请号 MYPI9902848 申请日期 1999.07.07
申请人 IPSEN PHARMA S.A.S. 发明人 PREVOST GREGOIRE;LONCHAMPT MARIE-ODILE;GORDON THOMAS
分类号 C07D233/64;C07D487/04;A61K31/198;A61K31/223;A61K31/4164;A61K31/421;A61K31/426;A61K31/495;A61K31/496;A61K31/4985;A61P3/04;A61P3/06;A61P3/10;A61P5/00;A61P9/12;A61P15/00;A61P25/02;A61P25/28;A61P31/12;A61P35/00;A61P37/02;C07D241/04;C07D263/32;C07D277/28;C07D417/06;C12N9/88 主分类号 C07D233/64
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