| 发明名称 |
Method of preparing alkylated salicylamides via a dicarboxylate intermediate |
| 摘要 |
The present invention relates to a method of preparing an alkylated salicylamide from a protected and activated salicylamide via a dicarboxylated salicylamide intermediate. The present invention also relates to dicarboxylic salicylamide delivery agent compounds for the delivery of active agents. Methods of administration are provided as well.
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| 申请公布号 |
US2006084646(A1) |
申请公布日期 |
2006.04.20 |
| 申请号 |
US20050040612 |
申请日期 |
2005.01.19 |
| 申请人 |
EMISPHERE TECHNOLOGIES, INC. |
发明人 |
BERNADINO JOSEPH N.;O'TOOLE DORIS C.;BAY WILLIAM E. |
| 分类号 |
A61K31/538;C07D265/36;A61K31/195;A61K45/00;A61K47/16;A61P1/04;A61P3/00;A61P3/02;A61P5/06;A61P7/00;A61P7/02;A61P9/00;A61P9/08;A61P9/12;A61P11/06;A61P13/00;A61P15/00;A61P19/08;A61P19/10;A61P31/00;A61P35/00;A61P37/02;A61P37/08;A61P43/00;C07C231/12;C07C235/60;C07C235/70;C07C269/00;C07C271/64;C07D265/12;C07D265/22;C07D265/26 |
主分类号 |
A61K31/538 |
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