发明名称 EFFICIENT SYNTHESIS OF 4,5-DIHYDRO-PYRAZOLO[3,4-C]PYRID-2-ONES
摘要 A novel process and intermediates thereof for making 4,5-dihydro-pyrazolo[3,4-c]pyrid-2-ones of the type shown below from appropriate phenyl hydrazines is described. Formula (I). These compounds can be useful as factor Xa inhibitors.
申请公布号 WO2006036926(A2) 申请公布日期 2006.04.06
申请号 WO2005US34511 申请日期 2005.09.27
申请人 BRISTOL-MYERS SQUIBB COMPANY;MUDRYK, BOGUSLAW, M.;CUNIERE, NICOLAS;HSIEH, DAU-MING;ROSSANO, LUCIUS;LIANG, JING;CHEN, BANG-CHI;ZHANG, HUIPING;ZHAO, RULIN;WANG, BEI;DAVID, ADRIAN 发明人 MUDRYK, BOGUSLAW, M.;CUNIERE, NICOLAS;HSIEH, DAU-MING;ROSSANO, LUCIUS;LIANG, JING;CHEN, BANG-CHI;ZHANG, HUIPING;ZHAO, RULIN;WANG, BEI;DAVID, ADRIAN
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