发明名称 ANTIBACTERIAL AND ANTIFOULING OXATHIAZINES AND THEIR OXIDES
摘要 Use of 3-aryl-5,6-dihydro-1,4,2-oxathiazines and their oxides having formula (1), wherein n is 0, 1 or 2; R1 is hydrogen, C1-4alkyl or benzyl; and R represents (a) phenyl; phenyl substituted with 1 to 3 substituents independently selected from hydroxyl, halo, C1-12alkyl, C5-6cycloalkyl, trihalomethyl, phenyl, C1- 5alkoxy, C1-5alkylthio, tetrahydropyranyloxy, phenoxy, C1-4alkylcarbonyl, phenylcarbonyl, C1-4alkylsulfinyl, C1- 4alkylsulfonyl, carboxy or its alkali metal salt, C1-4alkyloxycarbonyl, C1- 4alkylaminocarbonyl, phenylaminocarbonyl, tolylaminocarbonyl, morpholinocarbonyl, amino, nitro cyano, dioxolanyl or C1-4alkyloxyiminomethy l; naphthyl; pyridinyl; thienyl, preferably when n is not 2; furanyl; or thienyl or furanyl substituted with one to three substituents independently selected from C1-4alkyl, C1-4alkyloxy, C1- 4alkylthio, halo, cyano, formyl, acetyl, benzoyl, nitro, C1-4alkyloxycarbony l, phenyl, phenylaminocarbonyl and C1-4alkyloxyiminomethyl; or R represents a radical of formula (b) wherein X is oxygen or sulfur; Y is nitrogen, CH or C(C1-4alkyloxy); and R" is hydrogen or C1-4alkyl, as an antibacterial, anti-yeast, antifungal, algicidal, anti- crustacean, molluscicidal ail general antifouling agent and compositions containing the same.
申请公布号 CA2168357(C) 申请公布日期 2006.03.21
申请号 CA19942168357 申请日期 1994.08.24
申请人 JANSSEN PHARMACEUTICA NAAMLOZE VENNOOTSCHAP 发明人 VAN GESTEL, JOZEF FRANS ELISABETHA
分类号 A01N43/88;C07D291/06;C07D419/04;C09D5/16 主分类号 A01N43/88
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