发明名称 MODULATORS OF NUCLEAR RECEPTORS
摘要 Compounds of the invention, such as compounds of formula (I), where n, m, A, R1, R2, R3, R4 and R5 are defined herein, are useful as modulators of the activity of liver X receptors. Pharmaceutical compositions containing the compounds and methods of using the compounds are also disclosed.
申请公布号 WO2006025979(A2) 申请公布日期 2006.03.09
申请号 WO2005US26353 申请日期 2005.07.24
申请人 EXELIXIS, INC.;BAYNE, CHRISTOPHER, D.;JOHNSON, ALAN, T.;LU, SHAO-PO;MOHAN, RAJU;NYMAN, MICHAEL, C.;SCHWEIGER, EDWIN, J.;STEVENS, WILLIAM, C., JR.;WANG, HAIXIA;XIE, YINONG;BANNEN, LYNNE, CANNE;CHAN, DIVA, SZE-MING;HUANG, PING;JAMMALAMADAKA, VASU;KHOURY, RICHARD, G.;MAC, MORRISON, B.;PARKS, JASON, JEVIOUS;WANG, YONG;XU, WEI 发明人 BAYNE, CHRISTOPHER, D.;JOHNSON, ALAN, T.;LU, SHAO-PO;MOHAN, RAJU;NYMAN, MICHAEL, C.;SCHWEIGER, EDWIN, J.;STEVENS, WILLIAM, C., JR.;WANG, HAIXIA;XIE, YINONG;BANNEN, LYNNE, CANNE;CHAN, DIVA, SZE-MING;HUANG, PING;JAMMALAMADAKA, VASU;KHOURY, RICHARD, G.;MAC, MORRISON, B.;PARKS, JASON, JEVIOUS;WANG, YONG;XU, WEI
分类号 A61K31/4439;C07D213/85;C07D401/04;C07D401/06;C07D401/12;C07D405/04;C07D405/06;C07D405/12;C07D409/04;C07D413/06;C07D417/04;C07D417/06;C07D417/12 主分类号 A61K31/4439
代理机构 代理人
主权项
地址