发明名称 |
LABELED SUBSTRATE CONJUGATES FOR IDENTIFYING ENZYME INHIBITORS |
摘要 |
<p>This invention provides labeled-substrate conjugates for assaying enzymes, particularly neuraminidases. Also provided are assays that are useful for identifying compounds that inhibit sialyltransferases or neuraminidases and may be useful in treating subjects with influenza. In particular, the present invention relates to methods of using such labeled substrate conjugates to screen for enzyme inhibitors, particularly in a high-throughput format.</p> |
申请公布号 |
WO2006025983(A2) |
申请公布日期 |
2006.03.09 |
申请号 |
WO2005US26437 |
申请日期 |
2005.07.25 |
申请人 |
THE REGENTS OF THE UNIVERSITY OF CALIFORNIA;YING, LAIQIANG;GERVAY-HAGUE, JACQUELYN |
发明人 |
YING, LAIQIANG;GERVAY-HAGUE, JACQUELYN |
分类号 |
C12Q1/48;C08B37/00 |
主分类号 |
C12Q1/48 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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