| 发明名称 |
VERFAHREN ZUR HERSTELLUNG VON AZA-MAKROLIDEN MIT 4(R)-NH2 |
| 摘要 |
The subject-matter of the invention is a process for the stereoselective preparation of a compound of general formula I by stereoselective displacement by a nitrogenous nucleophilic compound of the activated alcohol functional group present at this 4'' position in a corresponding derivative of formula II. |
| 申请公布号 |
DE60014849(T2) |
申请公布日期 |
2006.03.09 |
| 申请号 |
DE2000614849T |
申请日期 |
2000.01.17 |
| 申请人 |
MERIAL, LYON |
发明人 |
LEON, PATRICK;LHERMITTE, FREDERIC;GUEVEL, RONAN;PAUZE, DENIS;GAREL, LAURENT;ODDON, GILLES |
| 分类号 |
A61K31/70;A61P31/00;C07B61/00;C07H17/08 |
主分类号 |
A61K31/70 |
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