发明名称 STABLE CRYSTAL FORM OF IMATINIB MESYLATE AND PROCESS FOR THE PREPARATION THEREOF
摘要 <p>The invention relates to a stable, non hygroscopic alpha crystalline form of methane sulfonic acid addition salt of 4-(4-methyl piperazin-lyl methyl)-N-[4-methyl-3-(4-pyridin-3-yl) pyrimidin-2-yl amino) phenyl]-benzamide (imatinib mesylate). A process for the preparation of the crystalline form is also described.</p>
申请公布号 WO2006024863(A1) 申请公布日期 2006.03.09
申请号 WO2005GB03392 申请日期 2005.09.02
申请人 CIPLA LIMITED;WAIN, CHRISTOPHER, PAUL;PATHI, SRINIVAS, LAXMINARAYAN;PUPPALA, RAVIKUMAR;KANKAN, RAJENDRA, NARAYANRAO;RAO, DHARMARAJ, RAMCHANDRA 发明人 PATHI, SRINIVAS, LAXMINARAYAN;PUPPALA, RAVIKUMAR;KANKAN, RAJENDRA, NARAYANRAO;RAO, DHARMARAJ, RAMCHANDRA
分类号 C07D401/14;A61K31/506;A61P35/00 主分类号 C07D401/14
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