发明名称 PYRROLO[2,3-d]PYRIMIDINES THAT MODULATE ACK1 AND LCK ACTIVITY
摘要 Compounds that modulate the action of ACK1 and LCK, and related compositions methods for treating ACK1- and LCK-mediated diseases are described. In one aspect, the compounds have the general structure: where the values of the substituents are provided herein.
申请公布号 WO2006004703(A3) 申请公布日期 2006.03.09
申请号 WO2005US22836 申请日期 2005.06.29
申请人 AMGEN INC.;FARTHING, CHRISTOPHER N.;FAULDER, PAUL;FRENKEL, ALEXANDER DAVID;HARRISON, MARTIN JAMES;JIAO, XIANYUN;KAYSER, FRANK;KOPECKY, DAVID J.;LIU, JINQIAN;LIVELY, SARAH E.;SHARMA, RAJIV;SHUTTLEWORTH, STEPHEN JOSEPH 发明人 FARTHING, CHRISTOPHER N.;FAULDER, PAUL;FRENKEL, ALEXANDER DAVID;HARRISON, MARTIN JAMES;JIAO, XIANYUN;KAYSER, FRANK;KOPECKY, DAVID J.;LIU, JINQIAN;LIVELY, SARAH E.;SHARMA, RAJIV;SHUTTLEWORTH, STEPHEN JOSEPH
分类号 C07D487/00;A61K31/519;A61P35/00 主分类号 C07D487/00
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