发明名称 DIARYLSULFONES AS 5-HT2A ANTAGONISTS
摘要 <p>Compounds of formula (I) are potent and selective antagonists of the human 5-HT2A receptor, and hence useful in treatment of a variety of adverse conditions of the CNS.</p>
申请公布号 WO2006021805(A1) 申请公布日期 2006.03.02
申请号 WO2005GB03352 申请日期 2005.08.26
申请人 MERCK SHARP & DOHME LIMITED;CASTRO PINEIRO, JOSE, LUIS;COOPER, LAURA, CATHERINE;GILLIGAN, MYRA;HUMPHRIES, ALEXANDER, CHARLES;HUNT, PETER, ALAN;LADDUWAHETTY, TAMARA;MACLEOD, ANGUS, MURRAY;MERCHANT, KEVIN, JOHN;VAN NIEL, MONIQUE, BODIL;WILSON, KEVIN 发明人 CASTRO PINEIRO, JOSE, LUIS;COOPER, LAURA, CATHERINE;GILLIGAN, MYRA;HUMPHRIES, ALEXANDER, CHARLES;HUNT, PETER, ALAN;LADDUWAHETTY, TAMARA;MACLEOD, ANGUS, MURRAY;MERCHANT, KEVIN, JOHN;VAN NIEL, MONIQUE, BODIL;WILSON, KEVIN
分类号 C07C317/14;C07C317/22;C07C317/24;C07C317/28;C07C317/32;C07C317/36;C07C317/42;C07C317/44;C07D205/04;C07D207/10;C07D211/38;C07D211/72;C07D213/34;C07D213/71;C07D217/24;C07D231/12;C07D233/54;C07D241/08;C07D249/08;C07D261/08;C07D271/10;C07D277/26;C07D295/096;C07D317/62;C07D319/18;(IPC1-7):C07C317/44;A61K31/10;C07D233/64;A61K31/416;A61K31/419;A61K31/397;A61K31/277 主分类号 C07C317/14
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