发明名称 Anhydrous crystalline azido cytosine hemisulfate derivative.
摘要 The present invention relates to the hemisulfate salt of 4-amino-1-((2r,3r,4s,5r)-5-azido-3,4-dihydroxy-5-hydroxymethyl-tetrahydro-furan-2-yl)-1h-pyrimidin-2-one with improved stability and physical properties which facilitate manufacturing, handling and formulating I and polymorphic crystalline forms thereof.
申请公布号 ZA200504472(B) 申请公布日期 2006.02.22
申请号 ZA20050004472 申请日期 2005.05.31
申请人 F. HOFFMANN-LA ROCHE AG 发明人 TERRENCE JOSEPH CONNOLLY;ANTHONY PRINCE;MARTIN JOSEPH ARMSTRONG;KESHAB SARMA
分类号 A61K31/70;A61K31/7052;A61K31/7068;A61K31/7072;A61P31/12;C07H19/06;C07H19/067 主分类号 A61K31/70
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