发明名称 |
1-(1, 2-Disubstituted piperidinyl)-4-substituted piperidine derivative, process for its preparation, pharmaceutical composition in which the derivative is comprised as well as process for its preparation |
摘要 |
<p>1-(1,2-Disubstituovaný piperidyl)-4-substituovanýderivát piperidinu, kde jednotlivé symboly mají specifický význam, jeho N-oxidová forma, farmaceuticky prijatelná adicní sul a stereochemicky izomerní forma. Zpusob jeho prípravy a pouzití, farmaceutický prostredek s jeho obsahem a zpusob jeho prípravy. Deriváty vzorce I jsou antagonisty substance P.</p> |
申请公布号 |
CZ296316(B6) |
申请公布日期 |
2006.02.15 |
申请号 |
CZ19980001864 |
申请日期 |
1996.12.20 |
申请人 |
JANSSEN PHARMACEUTICA N. V. |
发明人 |
JANSSENS FRANS EDUARD;SOMMEN FRANþOIS MARIA;SURLERAUX DOMINIQUE LOUIS NESTOR GHISLAINE;VAN ROOSBROECK YVES EMIEL MARIA |
分类号 |
C07D211/44;A61K31/00;A61K31/4427;A61K31/443;A61K31/4433;A61K31/445;A61K31/4465;A61K31/4523;A61K31/454;A61K31/4545;A61K31/47;A61K31/4709;A61K31/495;A61K31/4965;A61K31/497;A61K31/498;A61K31/505;A61K31/506;A61P43/00;C07D211/46;C07D211/52;C07D211/58;C07D401/06;C07D401/14;C07D405/14;C07D409/14;C07D417/14;C07D471/10;C07D491/10;C07D491/113 |
主分类号 |
C07D211/44 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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