发明名称 |
PROCESS FOR THE PREPARATION OF RACEMIC 2-[[2-(4-HYDROXYPHENYL)ETHYL]THIO]-3-[4-(2-[4-[(METHYLSULFONYL)OXY]PHENOXY]ETHYL)PHENYL]-PROPANOIC ACID |
摘要 |
The present invention provides a process for the preparation of substantially racemic 2-{[2-(4-hydroxyphenyl)ethyl]thio}-3-[4-(2-{4- [(methylsulfonyl)oxy]phenoxy}ethyl)phenyl]-propanoic acid which comprises reacting 2-{[2-(4-hydroxyphenyl)ethyl]thio}-3-[4-(2-{4-[(methylsulfonyl) oxy]phenoxy}ethyl)phenyl]propanoic acid enriched in one enantiomer with a base in an inert solvent.
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申请公布号 |
KR20060010840(A) |
申请公布日期 |
2006.02.02 |
申请号 |
KR20057024130 |
申请日期 |
2005.12.16 |
申请人 |
ASTRAZENECA AB |
发明人 |
ANDERSSON KJELL;LINDSTEDT ALSTERMARK EVA LOTTE;SORENSEN HENRIK |
分类号 |
C07C319/20;A61K31/192;C07C323/56;C07F7/18 |
主分类号 |
C07C319/20 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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