发明名称 NEW PSEUDOPOLYMORPH OF DESLORATADINE FORMED WITH CARBON DIOXIDE
摘要 The pseudopolymorph of desloratadine formed with carbon dioxide of the formula (I) has valuable anti-allergic effect and can be used as pharmaceutical active ingredient. The present invention also relates to the preparation of desloratadine of high purity. The present invention also relates to the use of the pseudopolymorph of desloratadine of the formula (I) for the preparation of salts of desloratadine of the formula (VI) (wherein X stands for an anion and n is 1 or 2).
申请公布号 WO2006003479(A2) 申请公布日期 2006.01.12
申请号 WO2005HU00073 申请日期 2005.07.07
申请人 EGIS GYOGYSZERGYAR RT.;MEZEI, TIBOR;SIMIG, GYULA;LUKACS, GYULA;PORCS-MAKKAY, MARTA;VOLK, BALAZS;MOLNAR, ENIKO;HOFMANNE FEKETE, VALERIA;SZENT-KIRALLYI, ZSUZSANNA 发明人 MEZEI, TIBOR;SIMIG, GYULA;LUKACS, GYULA;PORCS-MAKKAY, MARTA;VOLK, BALAZS;MOLNAR, ENIKO;HOFMANNE FEKETE, VALERIA;SZENT-KIRALLYI, ZSUZSANNA
分类号 C07D407/04;A61K31/352 主分类号 C07D407/04
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