发明名称 CONTRAST AGENTS ENDOWED WITH HIGH RELAXIVITY
摘要 The present invention relates to a novel class of paramagnetic ion-based contrast agents of formula (I), wherein a chelating backbone moiety is highly functionalized by the presence of one or more polyhdroxylated chain, that show a pharmacokinetic profile analogous to that of the commonly used T1-general extravascular agents (NSA) but are further characterized by a higher relaxivity.
申请公布号 WO2006002873(A2) 申请公布日期 2006.01.12
申请号 WO2005EP06956 申请日期 2005.06.28
申请人 BRACCO IMAGING SPA;AIME, SILVIO;GALLI, MATTEO;LATTUADA, LUCIANO;MOROSINI, PIERFRANCESCO;UGGERI, FULVIO;KONDAREDDIAR, RAMALINGAM 发明人 AIME, SILVIO;GALLI, MATTEO;LATTUADA, LUCIANO;MOROSINI, PIERFRANCESCO;UGGERI, FULVIO;KONDAREDDIAR, RAMALINGAM
分类号 A61K49/00;A61K49/06;A61K49/10;C07C229/76;C07D233/02;C07D257/02;C07D401/14;C07D405/14;C07F9/02 主分类号 A61K49/00
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