发明名称 |
PROCESS FOR PRODUCING ENANTIOPURE BETA-AMINO ACID DERIVATIVES, AND ENANTIOPURE BETA-AMINO ACID DERIVATIVES |
摘要 |
<p>Process for producing enantiopure beta-amino acid derivatives corresponding to general formula (I) R1-NZ-CHR2-CH2-COOR3 (I) in which R1 and R2 independently denote organic residues optionally forming a cyclic substituent, R3 denotes H or an organic residue, and Z represents H or an amino function-protecting group, comprising a step in which a mixture of enantiomers of a compound corresponding to general formula (II) R1-NZ-CHR2-CH2-COOR4 (II) in which R1, R2 and Z are as defined for formula (I), and R4 is an organic residue, is subjected to hydrolysis in the presence of a lipase.</p> |
申请公布号 |
EP1613762(A2) |
申请公布日期 |
2006.01.11 |
申请号 |
EP20040725376 |
申请日期 |
2004.04.02 |
申请人 |
SOLVAY (SOCIETE ANONYME) |
发明人 |
CALLENS, ROLAND;LARCHEVEQUE, MARC;POUSSET, CYRILLE |
分类号 |
C07D207/08;C07D265/30;C12P13/04;C12P17/14;C12P41/00;(IPC1-7):C12P41/00;C07K1/00 |
主分类号 |
C07D207/08 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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