发明名称 |
SUBSTITUTED PIPERIDINE DERIVATIVES, PHARMACEUTICAL COMPOSITIONS CONTAINING THE SAME AND USE THEREOF AS ANTIPSYCHOTIC AND ANALGESIC AGENTS |
摘要 |
<p>The invention relates to the following piperidine derivatives: 1-4-[3-[4-(6-flouro-1,2-benzisoxazol-3-yl)-1-piperidinyl]propoxy-3-methoxy-phenyl]-2-hydroxyethanone or a corresponding pharmaceutically acceptable acid addition salt, 4-[3-[4-(6-fluoro-1,2-benzisoxazol-3-yl)-1-piperidinyl]propoxy]-2-hydroxy-5-methoxy-alpha-methylbenzene-methanol or a corresponding pharmaceutically acceptable acid addition salt and 1-4-[3-[4-fluoro-1,2-benzisoxazol-3-yl)-1-piperidinyl]propoxy]-2-hydroxy-5-methoxyphenyl]ethanone or a corresponding pharmaceutically acceptable acid addition salt, to antipsychotic, analgesic and depot pharmaceutical compositions comprising said compounds and to the use thereof as antipsychotic or analgesic agents.</p> |
申请公布号 |
RO120341(B1) |
申请公布日期 |
2005.12.30 |
申请号 |
RO19960000888 |
申请日期 |
1994.10.27 |
申请人 |
HOECHST ROUSSEL PHARMACEUTICALS INC. |
发明人 |
STRUPCZEWSKI JOSEPH;HELSLEY C. GROVER;GLAMKOWSKI J. EDWARD;CHIANG YULIN;BORDEAU J. KENNETH;NEMOTO PETER A.;TEGELER JOHN J. |
分类号 |
A61K31/415;A61K31/42;A61K31/425;A61K31/44;A61K31/4427;A61K31/445;A61K31/4453;A61K31/47;A61K31/495;A61K31/496;A61K31/505;A61K31/55;A61P23/00;A61P25/00;A61P25/04;A61P25/18;C07C45/45;C07C45/67;C07C45/71;C07C49/84;C07C233/25;C07C233/33;C07C255/54;C07C323/22;C07D207/08;C07D221/04;C07D231/56;C07D239/02;C07D261/20;C07D275/04;C07D275/06;C07D277/82;C07D401/00;C07D401/04;C07D401/12;C07D401/14;C07D403/00;C07D403/04;C07D403/12;C07D403/14;C07D405/04;C07D413/04;C07D413/12;C07D413/14;C07D417/00;C07D417/04;C07D417/14;C07D419/00;C07D471/04;C07F7/18;(IPC1-7):C07D417/04 |
主分类号 |
A61K31/415 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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