发明名称 |
Azaindole derivatives as inhibitors of p38 kinase |
摘要 |
The invention is directed to methods to inhibit p38 kinase, preferably p38-alpha using compounds which are azaindoles wherein the azaindoles are coupled through a piperidine or piperazine type linker to another cyclic moiety.
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申请公布号 |
US2005288299(A1) |
申请公布日期 |
2005.12.29 |
申请号 |
US20050107027 |
申请日期 |
2005.04.15 |
申请人 |
MAVUNKEL BABU J;PERUMATTAM JOHN J;LU QING;DUGAR SUNDEEP;GOYAL BINDU;WANG DAN X;CHAKRAVARTY SARVAJIT;LUEDTKE GREGORY R;NASHASHIBI IMAD;TESTER RICHLAND;TAN XUEFEI |
发明人 |
MAVUNKEL BABU J.;PERUMATTAM JOHN J.;LU QING;DUGAR SUNDEEP;GOYAL BINDU;WANG DAN X.;CHAKRAVARTY SARVAJIT;LUEDTKE GREGORY R.;NASHASHIBI IMAD;TESTER RICHLAND;TAN XUEFEI |
分类号 |
A61K31/496;A61K31/56;A61K39/395;A61K45/06;C07D471/04;(IPC1-7):A61K31/496;A61K31/454;C07D487/02;C07D43/02 |
主分类号 |
A61K31/496 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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