发明名称 Azaindole derivatives as inhibitors of p38 kinase
摘要 The invention is directed to methods to inhibit p38 kinase, preferably p38-alpha using compounds which are azaindoles wherein the azaindoles are coupled through a piperidine or piperazine type linker to another cyclic moiety.
申请公布号 US2005288299(A1) 申请公布日期 2005.12.29
申请号 US20050107027 申请日期 2005.04.15
申请人 MAVUNKEL BABU J;PERUMATTAM JOHN J;LU QING;DUGAR SUNDEEP;GOYAL BINDU;WANG DAN X;CHAKRAVARTY SARVAJIT;LUEDTKE GREGORY R;NASHASHIBI IMAD;TESTER RICHLAND;TAN XUEFEI 发明人 MAVUNKEL BABU J.;PERUMATTAM JOHN J.;LU QING;DUGAR SUNDEEP;GOYAL BINDU;WANG DAN X.;CHAKRAVARTY SARVAJIT;LUEDTKE GREGORY R.;NASHASHIBI IMAD;TESTER RICHLAND;TAN XUEFEI
分类号 A61K31/496;A61K31/56;A61K39/395;A61K45/06;C07D471/04;(IPC1-7):A61K31/496;A61K31/454;C07D487/02;C07D43/02 主分类号 A61K31/496
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