发明名称 |
HIGHLY SELECTIVE NOVEL AMIDATION METHOD |
摘要 |
<p>The present invention provides an industrial production method with a short process having a high yield of an aliphatic cyclic carboxamide having carboxyl group, which comprises reacting functional group-selectively using an inexpensive condensing agent without protecting the carboxyl group by esterification, that is, reacting carboxylic acid anhydride obtained by reacting carboxylic acid and tertiary carboxylic acid halide with aliphatic cyclic secondary amine having carboxyl group.</p> |
申请公布号 |
WO2005121133(A1) |
申请公布日期 |
2005.12.22 |
申请号 |
WO2005JP11091 |
申请日期 |
2005.06.10 |
申请人 |
TAKEDA PHARMACEUTICAL COMPANY LIMITED;INAGAKI, ATSUSHI;SERA, MISAYO |
发明人 |
INAGAKI, ATSUSHI;SERA, MISAYO |
分类号 |
C07C51/06;C07C231/02;C07D267/14;C07D413/06;(IPC1-7):C07D413/06;A61P3/06;A61K31/553 |
主分类号 |
C07C51/06 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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