发明名称 FUSED HETEROCYCLIC DERIVATIVE, MEDICINAL COMPOSITION CONTAINING THE SAME, AND MEDICINAL USE THEREOF
摘要 A fused heterocyclic derivative represented by the general formula (I) (wherein R1 is hydrogen, OH, etc.; R2 is hydrogen, halogeno, or alkyl; R3 and R4 each is hydrogen, OH, halogeno, etc.; Q is alkylene, etc.; ring A is aryl or heteroaryl; and G is the group represented by the formula (G1) or (G2)), (G1) (G2) a pharmacologically acceptable salt of the derivative, or a prodrug of either. They have excellent inhibitory activity against human SGLT and are useful as preventive or therapeutic agents for diseases attributable to hyperglycemia, such as diabetes, postprandial hyperglycemia, impaired glucose tolerance, complications of diabetes, and obesity.
申请公布号 KR20050119179(A) 申请公布日期 2005.12.20
申请号 KR20057018698 申请日期 2004.03.24
申请人 KISSEI PHARMACEUTICAL CO., LTD. 发明人 FUSHIMI NOBUHIKO;YONEKUBO SHIGERU;MURANAKA HIDEYUKI;SHIOHARA HIROAKI;TERANISHI HIROTAKA;SHIMIZU KAZUO;ITO FUMIAKI;ISAJI MASAYUKI
分类号 A61K31/7036;A61K31/7042;A61K31/7048;A61K31/7056;A61K31/706;A61P3/04;A61P3/06;A61P3/10;A61P7/10;A61P9/04;A61P9/10;A61P9/12;A61P19/06;A61P43/00;C07H15/203;C07H17/00;C07H17/02;C07H17/04;(IPC1-7):C07H15/203;A61K31/703 主分类号 A61K31/7036
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