发明名称 Multicyclic compounds for use as melanin concentrating hormone antagonists in the treatment of obesity and diabetes
摘要 The present invention relates to a melanin concentrating hormone antagonist compound of formula I: (I); or a pharmaceutically acceptable salt, solvate, enantiomer or prodrug thereof useful in the treatment, prevention or amelioration of symptoms associated with obesity and related diseases.
申请公布号 US2005272718(A1) 申请公布日期 2005.12.08
申请号 US20050512986 申请日期 2005.04.28
申请人 AMMENN JOCHEN;GILLIG JAMES R;HEINZ LAWRENCE J;HIPSKIND PHILIP A;KINNICK MICHAEL D;LAI YEN-SHI;MORIN JOHN M;NIXON JAMES A;OTT CARSTEN;SAVIN KENNETH A;SCHOTTEN THEO;SLIEKER LAWRENCE J;SNYDER NANCY J;ROBERTSON MICHAEL A 发明人 AMMENN JOCHEN;GILLIG JAMES R.;HEINZ LAWRENCE J.;HIPSKIND PHILIP A.;KINNICK MICHAEL D.;LAI YEN-SHI;MORIN JOHN M.;NIXON JAMES A.;OTT CARSTEN;SAVIN KENNETH A.;SCHOTTEN THEO;SLIEKER LAWRENCE J.;SNYDER NANCY J.;ROBERTSON MICHAEL A.
分类号 A61K31/341;A61K31/381;A61K31/40;A61K31/4196;A61K31/42;A61K31/421;A61K31/422;A61K31/4245;A61K31/426;A61K31/428;A61K31/433;A61K31/4439;A61K31/454;A61K31/4709;A61K31/496;A61K31/497;A61K31/506;A61K31/5377;A61K31/541;A61K31/55;A61K31/551;A61P1/00;A61P1/04;A61P3/04;A61P3/06;A61P3/10;A61P5/06;A61P9/04;A61P9/10;A61P9/12;A61P11/06;A61P11/14;A61P13/02;A61P13/08;A61P15/12;A61P19/02;A61P25/08;A61P25/20;A61P25/22;A61P25/24;A61P25/28;A61P27/02;A61P29/00;A61P43/00;C07D207/333;C07D249/08;C07D261/08;C07D263/32;C07D271/06;C07D271/10;C07D271/107;C07D277/26;C07D285/12;C07D307/42;C07D333/18;C07D413/02;C07D413/04;C07D413/06;C07D413/10;C07D413/12;C07D413/14;C07D417/12;(IPC1-7):A61K31/55;A61K31/537;A61K31/424 主分类号 A61K31/341
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