发明名称 |
Multicyclic compounds for use as melanin concentrating hormone antagonists in the treatment of obesity and diabetes |
摘要 |
The present invention relates to a melanin concentrating hormone antagonist compound of formula I: (I); or a pharmaceutically acceptable salt, solvate, enantiomer or prodrug thereof useful in the treatment, prevention or amelioration of symptoms associated with obesity and related diseases.
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申请公布号 |
US2005272718(A1) |
申请公布日期 |
2005.12.08 |
申请号 |
US20050512986 |
申请日期 |
2005.04.28 |
申请人 |
AMMENN JOCHEN;GILLIG JAMES R;HEINZ LAWRENCE J;HIPSKIND PHILIP A;KINNICK MICHAEL D;LAI YEN-SHI;MORIN JOHN M;NIXON JAMES A;OTT CARSTEN;SAVIN KENNETH A;SCHOTTEN THEO;SLIEKER LAWRENCE J;SNYDER NANCY J;ROBERTSON MICHAEL A |
发明人 |
AMMENN JOCHEN;GILLIG JAMES R.;HEINZ LAWRENCE J.;HIPSKIND PHILIP A.;KINNICK MICHAEL D.;LAI YEN-SHI;MORIN JOHN M.;NIXON JAMES A.;OTT CARSTEN;SAVIN KENNETH A.;SCHOTTEN THEO;SLIEKER LAWRENCE J.;SNYDER NANCY J.;ROBERTSON MICHAEL A. |
分类号 |
A61K31/341;A61K31/381;A61K31/40;A61K31/4196;A61K31/42;A61K31/421;A61K31/422;A61K31/4245;A61K31/426;A61K31/428;A61K31/433;A61K31/4439;A61K31/454;A61K31/4709;A61K31/496;A61K31/497;A61K31/506;A61K31/5377;A61K31/541;A61K31/55;A61K31/551;A61P1/00;A61P1/04;A61P3/04;A61P3/06;A61P3/10;A61P5/06;A61P9/04;A61P9/10;A61P9/12;A61P11/06;A61P11/14;A61P13/02;A61P13/08;A61P15/12;A61P19/02;A61P25/08;A61P25/20;A61P25/22;A61P25/24;A61P25/28;A61P27/02;A61P29/00;A61P43/00;C07D207/333;C07D249/08;C07D261/08;C07D263/32;C07D271/06;C07D271/10;C07D271/107;C07D277/26;C07D285/12;C07D307/42;C07D333/18;C07D413/02;C07D413/04;C07D413/06;C07D413/10;C07D413/12;C07D413/14;C07D417/12;(IPC1-7):A61K31/55;A61K31/537;A61K31/424 |
主分类号 |
A61K31/341 |
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