发明名称 UREA ANTAGONISTS OF P2Y1 RECEPTOR USEFUL IN THE TREATMENT OF THROMBOTIC CONDITIONS
摘要 The present invention provides novel pyridyl or phenyl ureas and analogues thereof, which are selective inhibitors of the human P2Y1 receptor. The invention also provides for various pharmaceutical compositions of the same and methods for treating diseases responsive to modulation of P2Y1 receptor activity.
申请公布号 WO2005113511(A1) 申请公布日期 2005.12.01
申请号 WO2005US16422 申请日期 2005.05.11
申请人 BRISTOL-MYERS SQUIBB COMPANY;CHAO, HANNGUANG J.;TUERDI, HUJI;HERPIN, TIMOTHY;ROBERGE, JACQUES YVES;LIU, YALEI;LAWRENCE, R. MICHAEL;REHFUSS, ROBERT P.;CLARK, CHARLES G.;QIAO, JENNIFER X.;GUNGOR, TIMUR;LAM, PATRICK Y.S.;WANG, TAMMY C.;RUEL, REJEAN;L'HEUREUX, ALEXANDRE L.;THIBEAULT, CARL;BOUTHILLIER, GILLES;SCHNUR, DORA M. 发明人 CHAO, HANNGUANG J.;TUERDI, HUJI;HERPIN, TIMOTHY;ROBERGE, JACQUES YVES;LIU, YALEI;LAWRENCE, R. MICHAEL;REHFUSS, ROBERT P.;CLARK, CHARLES G.;QIAO, JENNIFER X.;GUNGOR, TIMUR;LAM, PATRICK Y.S.;WANG, TAMMY C.;RUEL, REJEAN;L'HEUREUX, ALEXANDRE L.;THIBEAULT, CARL;BOUTHILLIER, GILLES;SCHNUR, DORA M.
分类号 A61K31/4439;A61K31/444;A61K31/501;C07C275/30;C07C275/32;C07D213/40;C07D213/75;C07D213/89;C07D231/40;C07D231/50;C07D237/22;C07D333/36;C07D401/12;C07D401/14;C07D405/12;C07D405/14;C07D409/12;C07D409/14;C07D413/12;C07D417/12;C07F7/18 主分类号 A61K31/4439
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