发明名称 PROCESS FOR THE SYNTHESIS OF (IS)-4,5-DIMETHOXY-1-(METHYLAMINOMETHYL)-BENZOCYCLOBUTANE AND ADDITION SALTS THEREOF, AND TO THE APPLICATION THEREOF IN THE SYNTHESIS OF IVABRADINE AND ADDITION SALTS THEREOF WITH A PHARMACEUTICALLY ACCEPTABLE ACID
摘要 Process for the synthesis of the compound of formula (I): Application in the synthesis of ivabradine, addition salts thereof with a pharmaceutically acceptable acid, and hydrates thereof.
申请公布号 US2005261376(A1) 申请公布日期 2005.11.24
申请号 US20050060011 申请日期 2005.02.17
申请人 LERESTIF JEAN-MICHEL;BLANCO ISAAC G;LECOUVE JEAN-PIERRE;BRIGOT DANIEL 发明人 LERESTIF JEAN-MICHEL;BLANCO ISAAC G.;LECOUVE JEAN-PIERRE;BRIGOT DANIEL
分类号 C07D223/16;A61K31/55;A61P9/06;A61P9/10;C07B57/00;C07B61/00;C07C213/02;C07C213/08;C07C213/10;C07C217/56;C07C217/58;(IPC1-7):A61K31/137;C07C29/88 主分类号 C07D223/16
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