发明名称 |
PROCESS FOR THE SYNTHESIS OF (IS)-4,5-DIMETHOXY-1-(METHYLAMINOMETHYL)-BENZOCYCLOBUTANE AND ADDITION SALTS THEREOF, AND TO THE APPLICATION THEREOF IN THE SYNTHESIS OF IVABRADINE AND ADDITION SALTS THEREOF WITH A PHARMACEUTICALLY ACCEPTABLE ACID |
摘要 |
Process for the synthesis of the compound of formula (I): Application in the synthesis of ivabradine, addition salts thereof with a pharmaceutically acceptable acid, and hydrates thereof.
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申请公布号 |
US2005261376(A1) |
申请公布日期 |
2005.11.24 |
申请号 |
US20050060011 |
申请日期 |
2005.02.17 |
申请人 |
LERESTIF JEAN-MICHEL;BLANCO ISAAC G;LECOUVE JEAN-PIERRE;BRIGOT DANIEL |
发明人 |
LERESTIF JEAN-MICHEL;BLANCO ISAAC G.;LECOUVE JEAN-PIERRE;BRIGOT DANIEL |
分类号 |
C07D223/16;A61K31/55;A61P9/06;A61P9/10;C07B57/00;C07B61/00;C07C213/02;C07C213/08;C07C213/10;C07C217/56;C07C217/58;(IPC1-7):A61K31/137;C07C29/88 |
主分类号 |
C07D223/16 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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