| 发明名称 |
PROCESS FOR MAKING HIV PROTEASE INHIBITORS |
| 摘要 |
A process for making a compound of formula I comprises reacting an epoxide of formula IV with an amine of formula V, wherein R1, R2, R3, R4, r and a are defined herein. Compounds of formula I are useful as HIV protease inhibitors. <IMG>
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| 申请公布号 |
CA2167183(C) |
申请公布日期 |
2005.11.15 |
| 申请号 |
CA19942167183 |
申请日期 |
1994.07.11 |
| 申请人 |
MERCK & CO., INC. |
发明人 |
ASKIN, DAVID;VOLANTE, RALPH P.;ENG, KAN K. |
| 分类号 |
C07D263/52;C07D413/06;C07D453/02;C07D471/04;C07F9/653;(IPC1-7):C07D413/06 |
主分类号 |
C07D263/52 |
| 代理机构 |
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