发明名称 Crystalline 3-{4-methyl-3-[methyl-(7H-pyrrolo[2,3-d]pyrimidin-4-yl)-amino]-piperidin-1-yl}-3-oxo-propionitrile citrate
摘要 This invention relates to novel amorphous and crystallline forms of 3-{(3R,4R)-4-methyl-3-[methyl-(7H-pyrrolo[2,3-d]pyrimidin-4-yl)-amino]-piperidin-1-yl}-3-oxo-propionitrile mono citrate salt, useful as inhibitors of protein kinases, and to their methods of preparation.
申请公布号 US6965027(B2) 申请公布日期 2005.11.15
申请号 US20020310078 申请日期 2002.12.04
申请人 PFIZER INC. 发明人 FLANAGAN MARK E.;LI ZHENG J.
分类号 A61K31/519;A61K45/00;A61P1/04;A61P3/10;A61P11/06;A61P17/00;A61P17/06;A61P19/02;A61P25/00;A61P25/28;A61P29/00;A61P35/00;A61P35/02;A61P37/02;A61P37/06;A61P37/08;A61P43/00;C07D487/04;(IPC1-7):C07D401/12 主分类号 A61K31/519
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