发明名称 |
Nitrogen-containing heterocyclic compounds, their production and use |
摘要 |
A compound of the formula: wherein one of A and D is N and the other is C, or both are N; B is N or C; m is 0-3; R<SUP>1</SUP>, R<SUP>2 </SUP>and R<SUP>3 </SUP>each is (i) H or (ii) a group bound via C, N, O or S; R<SUP>4 </SUP>is a group bound via C; R<SUP>5 </SUP>is H or a group bound via C or O; R<SUP>6 </SUP>is H or a group bound via C; R<SUP>7 </SUP>is a homo- or hetero-cyclic group which may be substituted; or a salt thereof possesses excellent gonadotropin-releasing hormone antagonizing activity, and is useful as a prophylactic or therapeutic agent for sex hormone-dependent diseases, and so forth.
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申请公布号 |
US6962919(B2) |
申请公布日期 |
2005.11.08 |
申请号 |
US20020042229 |
申请日期 |
2002.01.11 |
申请人 |
TAKEDA PHARMACEUTICAL CO., LTD. |
发明人 |
FURUYA SHUICHI;IMAEDA TOSHIHIRO;SASAKI SATOSHI |
分类号 |
A61K31/506;A61P5/02;A61P15/18;C07D487/04;(IPC1-7):C07D239/70;A61K31/517;A61P5/06 |
主分类号 |
A61K31/506 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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