发明名称 |
Method for inhibiting p38 MAP kinase or TNF-alpha production using a 1,3-thiazole |
摘要 |
A 1,3-thiazole compound substituted at the 5-position by a pyridyl group optionally having substituent(s) has a superior p38 MAP kinase inhibitory activity and TNF-alpha production inhibitory activity.
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申请公布号 |
US6962933(B1) |
申请公布日期 |
2005.11.08 |
申请号 |
US20020048937 |
申请日期 |
2002.02.06 |
申请人 |
TAKEDA PHARMACEUTICAL COMPANY LIMITED |
发明人 |
OHKAWA SHIGENORI;NARUO KENICHI;KIMURA HIROYUKI;MIWATASHI SEIJI |
分类号 |
A61K31/4439;A61K31/444;A61P1/04;A61P3/10;A61P7/06;A61P7/08;A61P9/10;A61P11/00;A61P11/06;A61P19/02;A61P19/10;A61P21/00;A61P25/16;A61P25/28;A61P29/00;A61P31/06;A61P37/08;A61P39/02;A61P43/00;C07D417/04;C07D417/14;(IPC1-7):A61K31/442;A61K31/443 |
主分类号 |
A61K31/4439 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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