BENZAMIDE DERIVATIVES AS OXYTOCIN AGONISTS AND VASOPRESSIN ANTAGONISTS.

摘要

Novel compounds according to general formula 1, wherein Gl is NR5R6 or a fused polycyclic group that are specific OT receptor agonists and/or Vla receptor antagonists. Pharmaceutical compositions comprising such compounds are useful in the treatment of, inter alia, primary dysmenorrhoea.