发明名称 |
BENZYLPHOSPHATE AND SUBSTITUTED BENZYLPHOSPHATE PRODRUGS FOR THE TREATMENT OF PULMONARY INFLAMMATION |
摘要 |
A prodrug of a corticosteroid, lidocaine or related local anesthetic composition for formulation for delivery by aerosolization to inhibit inflammation in asthmatic lungs is described. The prodrug is preferably formulated in a 5 ml solution of a quarter normal saline having pH between 5.0 and 7.0 for the treatment of respiratory tract inflammation by an aerosol having mass medium average diameter predominantly between 1 to 5 µ produced by nebulization or dry powder inhaler.
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申请公布号 |
WO2005063777(A8) |
申请公布日期 |
2005.11.03 |
申请号 |
WO2004US42563 |
申请日期 |
2004.12.17 |
申请人 |
CORUS PHARMA;BAKER, WILLIAM, R.;STASIAK, MARCIN |
发明人 |
BAKER, WILLIAM, R.;STASIAK, MARCIN |
分类号 |
A61K9/00;A61K31/58;A61K31/661;C07F9/12;C07J71/00;(IPC1-7):C07F9/02 |
主分类号 |
A61K9/00 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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