发明名称 Process for preparing water soluble diterpenes and their applications
摘要 Aqueous solutions of diterpenes such as Forskolin, its congeners, analogs and derivatives, up to approximately 6% concentration, are prepared using suitably substituted cyclodextrin as a solubilizing agents. In the absence of cyclodextrin, some diterpenes such as Forskolin are soluble in water only to concentrations of about 0.001%. Such aqueous solutions find applications in topical and systemic use, as pharmaceutical, cosmeceutical, nutraceutical preparations containing diterpenes such as Forskolin and congeners.
申请公布号 US6960300(B2) 申请公布日期 2005.11.01
申请号 US20030605086 申请日期 2003.09.08
申请人 SAMI LABS LIMITED 发明人 MAJEED MUHAMMED;KUMAR ARVIND;NAGABHUSHANAM KALYANAM;PRAKASH SUBBALAKSHMI
分类号 A23L1/30;A61K9/00;A61K31/352;A61K45/06;A61K47/40;C07D311/92;(IPC1-7):B01D11/02;B01D37/00;A61K9/08 主分类号 A23L1/30
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