AGENT FOR CONTROLLING CHOLESTEROL HOMEOSTASIS-ASSOCIATED GENE TRANSCRIPTION ACTIVITY MEDIATED BY FXR ACTIVATION

摘要

It is intended to provide a preventive/remedy for hyperlipemia having an elevated efficacy. This object is achieved by using the following compound (1) having an FXR activity. wherein R1 represents a functional group selected from among hydrogen, acyl, alkyl and aryl; R2 represents a functional group selected from among hydrogen, alkyl and aryl; and R3 represents a functional group selected from among alkyl, alkynyl and alkenyl.