发明名称 SUBSTITUTED HETEROCYCLIC COMPOUNDS, PREPARATION METHOD THEREFOR AND PHARMACEUTICAL COMPOSITIONS CONTAINING THE SAME
摘要 <p>The invention relates to compounds of the formula (see Formula 1) in which: - A is a divalent radical selected from: A1) -O-CO- A2) -CH2-O-CO- A3) -O-CH2-CO- A4) -O-CH2-CH2- A5) -N(R1)-CO- A6) -N(R1)-CO-CO- A7) -N(R1)-CH2-CH2- A8) -O-CH2- in which: - R1 is a hydrogen or a (Cl-C4)-alkyl; and - Het is a nitrogen-containing heterocycle. APPLICATION: Neurokinin receptor antagonists.</p>
申请公布号 CA2211668(C) 申请公布日期 2005.09.20
申请号 CA19962211668 申请日期 1996.01.30
申请人 SANOFI 发明人 PROIETTO, VINCENZO;VAN BROECK, DIDIER;EMONDS-ALT, XAVIER;GROSSRIETHER, ISABELLE;GUEULE, PATRICK
分类号 C07D265/10;A61K31/38;A61K31/415;A61K31/416;A61K31/439;A61K31/44;A61K31/4427;A61K31/445;A61K31/451;A61K31/495;A61K31/496;A61K31/535;A61K31/5355;A61K31/5375;A61K31/5377;A61P1/04;A61P1/08;A61P1/12;A61P7/02;A61P9/10;A61P11/00;A61P11/06;A61P13/08;A61P13/10;A61P13/12;A61P17/00;A61P17/06;A61P17/16;A61P19/02;A61P25/16;A61P25/18;A61P25/20;A61P25/22;A61P25/24;A61P25/28;A61P25/30;A61P25/32;A61P27/02;A61P27/16;A61P29/00;A61P35/00;A61P37/08;A61P43/00;C07C215/28;C07C215/30;C07C217/08;C07C219/14;C07C219/22;C07C233/18;C07C255/03;C07C255/36;C07C255/42;C07C255/43;C07C271/20;C07C271/22;C07D209/10;C07D213/28;C07D213/36;C07D231/12;C07D263/10;C07D263/20;C07D263/38;C07D265/30;C07D265/32;C07D309/12;C07D333/10;C07D333/54;C07D401/06;C07D405/12;C07D413/06;C07D413/12;C07D413/14;C07D417/14;C07D453/02;(IPC1-7):C07D413/06;C07D241/08;C07D471/04;A61K31/55;A61K31/54;A61K31/435;C07D263/24;C07D409/14;C07D405/14;C07D401/14 主分类号 C07D265/10
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