发明名称 AMINO SUBSTITUTED DIARYL[A,D]CYCLOHEPTENE ANALOGS AS MUSCARINIC AGONISTS AND METHODS OF TREATMENT OF NEUROPSYCHIATRIC DISORDERS
摘要 Disclosed herein are analogs of clozapine and pharmaceutically acceptable salts, esters, amides, or prodrugs thereof; methods of synthesizing the analogs; and methods of using the analogs for treating neuorpsychiatric disorders. In some embodiments, the analogs are amino substituted diaryl[a,d]cycloheptenes.
申请公布号 WO2005063254(A3) 申请公布日期 2005.09.15
申请号 WO2004US43224 申请日期 2004.12.21
申请人 ACADIA PHARMACEUTICALS INC.;EK, FREDRIK;OLSSON, ROGER;OHLSSON, JOERGEN 发明人 EK, FREDRIK;OLSSON, ROGER;OHLSSON, JOERGEN
分类号 A61K31/55;A61K31/551;A61K31/553;A61K31/554;C07D403/04 主分类号 A61K31/55
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