摘要 |
The present invention can provide novel compounds useful as orally administrable growth hormone releaser, more specifically a benzimidazolidinone derivative of formula (1) or a pharmaceutically acceptable salt thereof: (1) wherein R<SUP>1 </SUP>is optionally substituted alkyl or the like; R<SUP>2</SUP>, R<SUP>3 </SUP>and R<SUP>4 </SUP>are each hydrogen, optionally substituted alkyl, or the like; R<SUP>5 </SUP>is optionally substituted aryl; q is 0 or 1; and W<SUP>1 </SUP>is a group represented by formula (2): (2) n is 1, 2 or 3; m is 0, 1, 2 or 3; R<SUP>6 </SUP>and R<SUP>7 </SUP>are each hydrogen, optionally substituted alkyl, or the like; and R<SUP>8 </SUP>and R<SUP>9 </SUP>are each hydrogen, optionally substituted alkyl, or the like.
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