| 发明名称 |
THE CITRATE SALT OF 5,8,14,-TRIAZATETRACYCLO(10.3.1.02,11.04,9)-HEXADECA-2(11),3,5,7,9-PENTAENE |
| 摘要 |
The present invention is directed to the citrate salt of 5,8,14-triazatetracyclo[10.3.1.0<2,11>.0<4,9>]-hexadeca-2(11),3,5,7,9-pentaene:and pharmaceutical compositions thereof. The present invention is also directed to the various forms of the citrate salt, particularly its hydrate and its anhydrous/nearly anhydrous polymorph. The invention is also directed to processes for preparation of these citrate salt forms. |
| 申请公布号 |
EP1390366(B1) |
申请公布日期 |
2005.08.31 |
| 申请号 |
EP20020724553 |
申请日期 |
2002.04.26 |
| 申请人 |
PFIZER PRODUCTS INC. |
发明人 |
JOHNSON, PHILIP, JAMES;ROSE, PETER, ROBERT;WINT, LEWIN, THEOPHILUS;WILLIAMS, GLENN, ROBERT |
| 分类号 |
C07D487/08;A61K;A61K31/495;A61K31/529;A61P;A61P1/04;A61P3/04;A61P5/14;A61P9/06;A61P9/12;A61P17/00;A61P17/02;A61P25/00;A61P25/04;A61P25/06;A61P25/08;A61P25/10;A61P25/14;A61P25/16;A61P25/18;A61P25/20;A61P25/22;A61P25/24;A61P25/28;A61P25/30;A61P25/32;A61P25/36;A61P27/00;A61P29/00;A61P31/18;A61P39/02;C07D;C07D221/00;C07D223/00;C07D471/08 |
主分类号 |
C07D487/08 |
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