发明名称 Amidinylphenyl compounds and their use as fungicides
摘要 Compounds of the formula (R<SUP>5</SUP>)<SUB>m</SUB>-(R<SUP>6</SUP>A)-2-(R<SUP>4</SUP>)-1-[N-C(R<SUP>1</SUP>)N(R<SUP>2</SUP>)(R<SUP>3</SUP>)]benzene and their agriculturally suitable salts, are disclosed which are useful as fungicides, wherein R<SUP>1 </SUP>is H, OH, SH, SO<SUB>3</SUB>H, CN, -OR<SUP>7 </SUP>or -SR<SUP>7</SUP>; C<SUB>1</SUB>-C<SUB>10 </SUB>alkyl, C<SUB>2</SUB>-C<SUB>10 </SUB>alkenyl, C<SUB>2</SUB>-C<SUB>5 </SUB>alkoxycarbonyl, C<SUB>2</SUB>-C<SUB>10 </SUB>alkynyl, a C<SUB>3</SUB>-C<SUB>6 </SUB>carbocycle or a 3-, 4-, 5- or 6-membered heterocycle, each optionally substituted; provided that when R<img id="custom-character-00001" he="2.46mm" wi="1.44mm" file="US20050182025A1-20050818-P00900.TIF" alt="custom character" img-content="character" img-format="tif"/>1? is a heterocycle containing nitrogen as a ring member, it is not attached to the remainder of Formula I through said nitrogen ring member; R<SUP>6 </SUP>is C<SUB>5</SUB>-C<SUB>21 </SUB>alkyl, C<SUB>5</SUB>-C<SUB>21 </SUB>alkenyl, C<SUB>5</SUB>-C<SUB>21 </SUB>alkynyl, C<SUB>4</SUB>-C<SUB>9</SUB>alkoxycarbonyl, C<SUB>4</SUB>-C<SUB>6 </SUB>alkylaminocarbonyl, C<SUB>3</SUB>-C<SUB>10 </SUB>dialkylaminocarbonyl or C<SUB>3</SUB>-C<SUB>12 </SUB>trialkylsilyl, each optionally substituted; or R<SUP>6 </SUP>is C<SUB>1</SUB>-C<SUB>4 </SUB>alkyl or C<SUB>2</SUB>-C<SUB>9 </SUB>alkylcarbonyl, each substituted with one or more R<SUP>12</SUP>; A is a direct bond, O, S(O)<SUB>n</SUB>, or NR<SUP>10</SUP>; n is 0, 1 or 2; m is 0, 1, 2 or 3; and R<SUP>2</SUP>, R<SUP>3</SUP>, R<SUP>4</SUP>, R<SUP>5</SUP>, R<SUP>7</SUP>, R<SUP>10 </SUP>and R<SUP>12 </SUP>are as defined in the disclosure. Also disclosed are compositions containing the compounds of the formula (R<SUP>5</SUP>)<SUB>m</SUB>-(R<SUP>6</SUP>A)-2-(R<SUP>4</SUP>)-1-[N-C(R<SUP>1</SUP>)N(R<SUP>2</SUP>)(R<SUP>3</SUP>)]benzene and a method for controlling plant diseases caused by fungal plant pathogens which involves applying an effective amount of a compound of the formula (R<SUP>5</SUP>)<SUB>m</SUB>-(R<SUP>6</SUP>A)-2-(R<SUP>4</SUP>)-1-[N-C(R<SUP>1</SUP>)N(R<SUP>2</SUP>)(R<SUP>3</SUP>)]benzene.
申请公布号 US2005182025(A1) 申请公布日期 2005.08.18
申请号 US20040510083 申请日期 2004.10.01
申请人 TSENG CHI-PING 发明人 TSENG CHI-PING
分类号 C07C257/12;A01N25/02;A01N25/08;A01N25/30;A01N37/52;A01N47/30;A01N47/42;A01N49/00;A01N55/00;C07C257/10;C07C257/14;C07C275/34;C07C275/70;C07C323/20;C07C323/36;C07C335/18;C07C335/36;C07F7/18;(IPC1-7):A01N55/00;A01N33/02;A01N43/40 主分类号 C07C257/12
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