发明名称 MACROCYCLIC COMPOUNDS USEFUL AS PHARMACEUTICALS
摘要 The present invention provides compounds having formula (I), and additionally provides methods for the synthesis thereof and methods for the use thereof in the treatment of various disorders including inflammatory or autoimmune disorders, and disorders involving malignancy or increased angiogenesis, wherein R 1 -R 11 , t, X, Y, Z and n are as defined herein.
申请公布号 PL373044(A1) 申请公布日期 2005.08.08
申请号 PL20030373044 申请日期 2003.03.07
申请人 EISAI CO LTD 发明人 BOIVIN ROCH;CHIBA KENICHI;DIEPITRO LUCIAN;DU HONG;EGUCHI YOSHIHITO;FUJITA MASANORI;GILBERT SANDRA;GOTO MASAKI;HARMANGE JEAN CHRISTOPHE;INOUE ATSUSHI;JIANG YIMIN;KAWADA MEGUMI;KAWAI TAKATOSHI;KAWAKAMI YOSHIYUKI;KIMURA AKIFUMI;KOTAKE MAKOTO;KUBOI YOSHIKAZU;LEMELIN CHARLES;LI XIANG-YI;MATSUSHIMA TOMOHIRO;MIZUI YOSHIHARU;SAKURAI HIDEKI;SHEN YONGCHUN;SPYVEE MARK;TANAKA ISAO;WANG YUAN;YAMAMOTO SATOSHI;YONEDA NAOKI;CHOW JESSE
分类号 C07D491/044;A61K31/335;A61K31/36;A61K31/365;A61K31/395;A61K31/4178;A61K31/4188;A61K31/5377;A61P1/00;A61P1/04;A61P1/16;A61P3/10;A61P7/04;A61P9/00;A61P9/10;A61P11/00;A61P11/02;A61P11/06;A61P17/00;A61P17/04;A61P17/06;A61P17/16;A61P19/02;A61P19/04;A61P19/10;A61P21/04;A61P25/00;A61P25/02;A61P25/08;A61P25/28;A61P27/02;A61P29/00;A61P31/04;A61P31/18;A61P33/06;A61P35/00;A61P37/02;A61P37/06;A61P37/08;A61P43/00;C07D267/00;C07D313/00;C07D401/12;C07D405/12;C07D491/04;C07D493/04;C07D521/00 主分类号 C07D491/044
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