发明名称 PHENYLALANINE DERIVATIVE
摘要 <p>Disclosed is a phenylalanine derivative having excellent VLA-4 inhibitory activity which is represented by the following general formula (1) or a salt thereof. (1) (In the formula, R&lt;1&gt; represents an aromatic hydrocarbon group having 6-10 carbon atoms or the like; Z represents a phenyl group or the like; R&lt;2&gt; represents a hydrogen atom or a lower alkyl group; n represents a number such as 0; and when n is 0, Y represents NOR&lt;3&gt; (wherein R&lt;3&gt; represents a methyl group or the like), CCl2 or the like.)</p>
申请公布号 WO2005068415(A1) 申请公布日期 2005.07.28
申请号 WO2005JP00666 申请日期 2005.01.20
申请人 FUJIYAKUHIN CO., LTD.;UDA, JUNICHIRO;OKAMOTO, YASUSHI;IWABUCHI, TAKEYUKI;INOUE, TSUTOMU;NAKANO, HIROYUKI;ISHIKAWA, TOMOHIKO;KAWASAKI, NOBUHIDE;KATOH, MASUMI 发明人 UDA, JUNICHIRO;OKAMOTO, YASUSHI;IWABUCHI, TAKEYUKI;INOUE, TSUTOMU;NAKANO, HIROYUKI;ISHIKAWA, TOMOHIKO;KAWASAKI, NOBUHIDE;KATOH, MASUMI
分类号 C07C233/51;C07C233/31;C07C233/49;C07C233/50;C07C251/38;C07C251/40;C07C251/42;C07C251/44;C07C251/48;C07C317/44;C07C323/59;C07C323/63;C07D209/20;C07D211/34;C07D213/56;C07D295/205;C07D307/54;C07D309/06;C07D317/60;C07D333/24;C07D335/02;C07D339/08;C07D409/12;(IPC1-7):C07C233/49;A61P43/00;A61P29/00;A61K31/537;A61K31/443;A61K31/440;A61K31/385;A61K31/382;A61K31/381;A61K31/351;A61K31/36;A61K31/341;A61K31/198;C07D417/04;C07D405/12;C07D333/22;C07D317/58;C07D295/20;C07D213/53;C07D211/06;C07D209/04;C07C317/50;C07C251/34 主分类号 C07C233/51
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