发明名称 PYRROLOTRIAZINE COMPOUNDS AS KINASE INHIBITORS
摘要 <p>The present invention provides compounds of formula (I); and pharmaceutically acceptable salts thereof. The formula (I) compounds inhibit tyrosine kinase activity of growth factor receptors such as HER1, HER2 and HER4 thereby making them useful as antiproliferative agents. The formula (I) compounds are also useful for the treatment of other diseases associated with signal transduction pathways operating through growth factor receptors.</p>
申请公布号 WO2005066176(A1) 申请公布日期 2005.07.21
申请号 WO2004US43169 申请日期 2004.12.23
申请人 BRISTOL-MYERS SQUIBB COMPANY;FINK, BRIAN, E.;GAVAI, ASHVINIKUMAR, V.;VITE, GREGORY, D.;CHEN, PING;MASTALERZ, HAROLD;NORRIS, DEREK, J.;TOKARSKI, JOHN, S.;ZHAO, YUFEN;HAN, WEN-CHING 发明人 FINK, BRIAN, E.;GAVAI, ASHVINIKUMAR, V.;VITE, GREGORY, D.;CHEN, PING;MASTALERZ, HAROLD;NORRIS, DEREK, J.;TOKARSKI, JOHN, S.;ZHAO, YUFEN;HAN, WEN-CHING
分类号 A61K31/53;C07D487/04;C07D519/00;(IPC1-7):C07D487/04;A61P35/00 主分类号 A61K31/53
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