发明名称 METHOD AND COMPOSITIONS FOR IDENTIFYING ANTI-HIV THERAPEUTIC COMPOUNDS
摘要 <p>Methods are provided for identifying anti-HIV therapeutic compounds substituted with carboxyl ester or phosphonate ester groups. Libraries of such compounds are screened optionally using the novel enzyme GS-7340 Ester Hydrolase. Compositions and methods relating to GS-7340 Ester Hydrolase also are provided.</p>
申请公布号 WO2005064008(A1) 申请公布日期 2005.07.14
申请号 WO2004US42991 申请日期 2004.12.22
申请人 GILEAD SCIENCES, INC.;ARIMILLI, MURTY N.;BECKER, MARK M.;BIRKUS, GABRIEL;BRYANT, CLIFFORD;CHEN, JAMES M.;CHEN, XIAOWU;CIHLAR, TOMAS;DASTGAH, AZAR;EISENBERG, EUGENE J.;FARDIS, MARIA 发明人 ARIMILLI, MURTY N.;BECKER, MARK M.;BIRKUS, GABRIEL;BRYANT, CLIFFORD;CHEN, JAMES M.;CHEN, XIAOWU;CIHLAR, TOMAS;DASTGAH, AZAR;EISENBERG, EUGENE J.;FARDIS, MARIA
分类号 C12N9/99;A61K31/4155;A61K31/66;A61K31/665;A61K31/675;A61P31/18;A61P43/00;C07D213/75;C07D213/85;C07D231/12;C07D231/20;C07D233/42;C07D239/48;C07D239/80;C07D243/04;C07D265/18;C07D307/68;C07D401/06;C07D403/06;C07D471/14;C07D491/04;C07F;C07F9/02;C07F9/38;C07F9/40;C07F9/44;C07F9/58;C07F9/62;C07F9/645;C07F9/6506;C07F9/6509;C07F9/6512;C07F9/653;C07F9/6533;C07F9/655;C07F9/6558;C07F9/6561;C07F9/6584;C12N9/16;C12Q1/18;C12Q1/37;C12Q1/44;C12Q1/70;G01N33/04;G01N33/50;(IPC1-7):C12Q1/44 主分类号 C12N9/99
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