发明名称 PROCESS FOR PRODUCTION OF VINYL PERFLUOROALKANESULFONATE DERIVATIVES
摘要 <CHEM> (wherein R<1>, R<2>, R<3>, R<4> and R<5> may be the same or different and each represents a hydrogen atom, substituted or unsubstituted lower alkyl, substituted or unsubstituted lower alkoxy, or the like; R<17> represents trifluoromethyl or the like; R<18>, R<19>, R<20>, R<21> and R<22> may be the same or different and each represents a hydrogen atom, substituted or unsubstituted lower alkyl, or the like). <??>An easy and simple process for producing a vinyl perfluoroalkanesulfonate derivative represented by general formula (IV) which is a useful intermediate in synthesis of medicines, natural products, or the like, at a low cost, is provided. The process is characterized by, for example, reacting a carbonyl compound represented by general formula (I) described above with a perfluoroalkanesulfonic anhydride represented by general formula (II) described above in the presence of a pyridine derivative represented by general formula (III) described above in an amount of 0.1 to 1.0 equivalent to the perfluoroalkanesulfonic anhydride.
申请公布号 EP1553082(A1) 申请公布日期 2005.07.13
申请号 EP20030760919 申请日期 2003.06.20
申请人 KYOWA HAKKO KOGYO CO., LTD. 发明人 KATO, SACHIKO;CHUJO, IWAO;SUZUKI, KOJI
分类号 C07C303/26;C07C309/65;C07J31/00;(IPC1-7):C07C303/26 主分类号 C07C303/26
代理机构 代理人
主权项
地址