发明名称 FUSED BENZENE DERIVATIVE AND USE
摘要 The present invention provides a compound represented by the general formula: <CHEM> Äwherein Ring A represents an optionally substituted 5- to 8-membered ring, Ring B represents a further optionally substituted 4- to 10-membered ring, Ring C represents a further optionally substituted benzene ring, X<1> represents carbon atom, X<2> represents a carbon atom, an oxygen atom, etc., W represents a nitrogen atom, etc., Y<11> represents a group represented by the formula CR<2>R<3'> (wherein R<2> represents a hydrogen atom, a cyano group, a nitro group, etc., and R<3'> represents a hydrogen atom, a cyano group, a nitro group, etc., respectively), Y<21> represents a group represented by the formula CR<4>R<5'> (wherein R<4> represents a hydrogen atom, a cyano group, a nitro group, etc., and R<5'> represents a hydrogen atom, a cyano group, a nitro group, etc., respectively), etc., and R<1> represents an electron-withdrawing group, respectively. The formula represents a single bond or a double bondÜ or a salt thereof, which is useful as an androgen receptor modulator.
申请公布号 EP1553074(A1) 申请公布日期 2005.07.13
申请号 EP20030788076 申请日期 2003.08.11
申请人 TAKEDA PHARMACEUTICAL COMPANY LIMITED 发明人 SHIRAISHI, MITSURU;HARA, TAKAHITO;KUSAKA, MASAMI;KANZAKI, NAOYUKI;YAMAMOTO, SATOSHI;MIYAWAKI, TOSHIO
分类号 A61P5/26;A61P13/08;A61P15/00;A61P15/10;A61P15/12;A61P19/10;A61P35/00;A61P43/00;C07C35/52;C07C217/04;C07C255/52;C07C255/53;C07C255/54;C07C255/56;C07D207/06;C07D207/08;C07D207/10;C07D207/12;C07D207/14;C07D207/16;C07D207/22;C07D207/24;C07D209/46;C07D211/22;C07D211/28;C07D211/34;C07D211/42;C07D211/46;C07D211/60;C07D211/62;C07D211/74;C07D231/08;C07D261/04;C07D265/02;C07D267/10;C07D295/073;C07D295/112;C07D295/155;C07D303/46;C07D307/79;C07D333/54;C07D405/04;C07D409/04;C07D491/10;C07D491/113;(IPC1-7):C07C35/52;C07D209/44;C07D211/14 主分类号 A61P5/26
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