发明名称 ЗАМЕЩЕННЫЕ ИНДАЗОЛЫ, ОБЛАДАЮЩИЕ ПРИТОВОРАКОВОЙ АКТИВНОСТЬЮ
摘要 Substituted indazoles (I), their salts, in non-chiral, racemic, or enantiomeric form and their mixtures, are new. Substituted indazoles (I), their salts, in non-chiral, racemic, or enantiomeric form and their mixtures, are new. R1 = H, halogen, alkyl, alkylene, alkynyl, aryl, heteroaryl, cycloalkyl, heterocyclo, substituted alkyl, substituted alkylene, substituted alkynyl, substituted aryl, substituted heteroaryl, substituted cycloalkyl, substituted heterocyclyl, CN, O(R2), OC(O)R2, OC(O)N(R2)(R3), OSO2(R2), N(R2)(R3), N=C(R2)(R3), N(R2)CO(R3), N(R4)CON(R2)(R3), N(R4)CSN(R2)(R3), N(R2)S(O2)(R3), COR2, COOR2, CON(R2)(R3), C(=N(R3))(R2), C(=N(OR3))(R2), SR2, SOR2, SO2R2, or SO2N(R2)(R3); R2, R3, and R4 = H, alkyl, aryl, cycloalkyl, heterocyclyl, substituted alkyl, substituted aryl, substituted cycloalkyl, substituted heterocyclyl, alkylene or substituted alkylene; X = SO2NH, SO2-O-, NHSO2, or O-SO2; Z = alkyl, aryl, heteroaryl, cycloalkyl, heterocyclyl, substituted alkyl, substituted aryl, substituted heteroaryl, substituted cycloalkyl, substituted heterocyclyl with the exception of the specific compounds defined below under Definitions.
申请公布号 RU2004130280(A) 申请公布日期 2005.06.27
申请号 RU20040130280 申请日期 2003.03.07
申请人 АВЕНТИС ФАРМА С.А. (FR) 发明人 ДАМУР Доминик (FR);КАРРИ Жан-Кристоф (FR);НЕМЕСЕК Патрик (FR);ТЕРРЬЕ Корин (FR);НАРДИ Фредерико (FR);ФИЛОШ Брюно (FR);ШЕРРЬЕ Мари-Пьер (FR);БЕЗАР Даниель (FR)
分类号 A61K31/416;A61K31/4184;A61K31/42;A61K31/4245;A61K31/437;A61K31/4439;A61K31/454;A61K31/695;A61P35/00;A61P43/00;C07D231/56;C07D401/04;C07D401/12;C07D403/04;C07D405/04;C07D409/04;C07D409/12;C07D413/12;C07D413/14;C07D471/04;C07F7/10 主分类号 A61K31/416
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