发明名称 TRIAZASPIRO[5.5]UNDECANE DERIVATIVES AND DRUGS COMPRISING THE SAME AS THE ACTIVE INGREDIENT
摘要 A compound represented by the following general formula (I): (I) wherein each symbol is as defined in the description; its quaternary ammonium salt, its N-oxide or a salt thereof. Compounds represented by the general formula (I) are useful in preventing and/or treating various inflammatory diseases (asthma, nephritis, nephropathy, hepatitis, arthritis, rheumatoid arthritis, rhinitis, conjunctivitis, ulcerative colitis, etc.), immune diseases (autoimmune disease, transplant rejection, immune suppression, psoriasis, multiple sclerosis, etc.), infection with human immunodeficiency virus (acquired immune deficiency syndrome), allergic diseases (atopic dermatitis, urticaria, allergic bronchopulmonary aspergillosis, allergic eosinophilic gastroenteritis, etc.), ischemic reperfusion injury, acute respiratory distress syndrome, shock accompanying bacterial infection, diabetes, cancer metastasis, etc.
申请公布号 KR20050057408(A) 申请公布日期 2005.06.16
申请号 KR20057004600 申请日期 2005.03.17
申请人 ONO PHARMACEUTICAL CO., LTD. 发明人 TAKAOKA YOSHIKAZU;NISHIZAWA RENA;SHIBAYAMA SHIRO;SAGAWA KENJI;MATSUO MASAYOSHI
分类号 A61P1/04;A61P1/16;A61P3/10;A61P9/00;A61P11/00;A61P11/02;A61P11/06;A61P13/12;A61P17/00;A61P17/06;A61P19/02;A61P25/00;A61P27/00;A61P29/00;A61P31/04;A61P31/18;A61P35/04;A61P37/02;A61P37/06;A61P37/08;A61P43/00;C07D471/10;(IPC1-7):C07D471/10 主分类号 A61P1/04
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