发明名称 |
TAXANE DERIVATIVES FUNCTIONALIZED AT THE 14- POSITION AND A PROCESS FOR THE PREPARATION THEREOF |
摘要 |
<p>A general process for the functionalization at the 14- position of 13-ketobaccatin derivatives of formula I to give derivatives of formula II
wherein the substituents are as defined in the disclosure. The conversion of compounds of formula II in compounds of formula III,
wherein the substituents are as defined in the disclosure, is also described.</p> |
申请公布号 |
EP1537093(A2) |
申请公布日期 |
2005.06.08 |
申请号 |
EP20030747971 |
申请日期 |
2003.09.05 |
申请人 |
INDENA S.P.A. |
发明人 |
FONTANA, GABRIELE;BOMBARDELLI, EZIO;BATTAGLIA, ARTURO;BALDELLI, ELEONORA;GUERRINI, ANDREA;GELMI, MARIA LUISA;CARENZI, GIACOMO;POCAR, DONATO |
分类号 |
C07D305/14;(IPC1-7):C07D305/14 |
主分类号 |
C07D305/14 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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