发明名称 |
CATHEPSIN CYSTEINE PROTEASE INHIBITORS |
摘要 |
This invention relates to class of compounds which are cysteine protease inhibitors, including but not limited to, inhibitors of cathepsins K, L, S and B. These compounds are useful for treating diseases in which inhibition of bone resorption is indicated, such as osteoporosis. They have the following structure: Formula (I) |
申请公布号 |
EP1537074(A1) |
申请公布日期 |
2005.06.08 |
申请号 |
EP20030793540 |
申请日期 |
2003.09.03 |
申请人 |
MERCK FROSST CANADA INC. |
发明人 |
BOYD, MICHAEL;GAGNON, MARC;LAU, CHEUK;MELLON, CHRISTOPHE;SCHEIGETZ, JOHN |
分类号 |
C07D295/08;A61K31/275;A61K31/381;A61K31/404;A61K31/4164;A61K31/426;A61K31/4409;A61K31/4439;A61K31/445;A61K31/47;A61K31/495;A61K31/497;A61K31/505;A61K31/5375;A61K31/69;A61K31/695;A61K45/00;A61P1/02;A61P3/14;A61P19/02;A61P19/08;A61P19/10;A61P35/00;A61P35/02;A61P43/00;C07C255/25;C07C255/29;C07C255/54;C07C259/10;C07C311/29;C07C317/22;C07C317/24;C07C317/44;C07C323/19;C07C323/22;C07C323/52;C07C323/60;C07D209/12;C07D211/20;C07D211/22;C07D211/94;C07D213/30;C07D213/61;C07D213/79;C07D213/89;C07D215/14;C07D215/60;C07D231/12;C07D233/22;C07D239/26;C07D241/16;C07D277/24;C07D295/088;C07D295/10;C07D295/192;C07D295/205;C07D295/26;C07D333/16;C07D401/04;C07F5/02 |
主分类号 |
C07D295/08 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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